Structural Effect on Adjuvanticity of Saponins

J Med Chem. 2020 Mar 26;63(6):3290-3297. doi: 10.1021/acs.jmedchem.9b02063. Epub 2020 Feb 26.

Abstract

We have prepared a number of saponin-based vaccine adjuvant candidates. These unnatural saponins have a different terminal-functionalized side chain incorporated into the glucuronic acid unit that is attached to a triterpenoid core at its C3 position. The semisynthetic saponin adjuvants have shown significantly different immunostimulatory activities, suggesting that the structure of the side chain, triterpenoid core, and oligosaccharide domain together orchestrate saponin adjuvant's potentiation of immune responses. Among these new adjuvant candidates, VSA-2 (5b), a derivative of Momordica saponin (MS) II, showed consistent enhancement of immunoglobulin G2a (IgG2a) production when it was in formulation with either ovalbumin or recombinant hemagglutinin B (rHagB) antigen. With rHagB antigen, it induced a significantly higher IgG2a response than the positive control GPI-0100, a well-studied semisynthetic saponin adjuvant mixture derived from Quillaja saponaria Molina saponins, known for its ability to induce a balanced Th1/Th2 immunity. These results confirm that Momordica saponins are a viable natural source to provide potent saponin adjuvants after simple chemical derivatization and identify VSA-2 (5b) as another MS-based promising immunostimulant lead owing to its distinctive ability in potentiating the IgG2a response.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adhesins, Bacterial / immunology
  • Adjuvants, Immunologic / chemical synthesis
  • Adjuvants, Immunologic / pharmacology*
  • Animals
  • Antibody Formation / drug effects
  • Chickens
  • Female
  • Immunoglobulin G / immunology
  • Immunoglobulin G / metabolism
  • Lectins / immunology
  • Mice, Inbred BALB C
  • Molecular Structure
  • Ovalbumin / immunology
  • Saponins / chemical synthesis
  • Saponins / immunology
  • Saponins / pharmacology*
  • Th1 Cells / drug effects

Substances

  • Adhesins, Bacterial
  • Adjuvants, Immunologic
  • GPI0100
  • HagB protein, Porphyromonas gingivalis
  • Immunoglobulin G
  • Lectins
  • Saponins
  • Ovalbumin